Eltoprazine hydrochloride, Catalog: B2301

Alternate Names 1-(2,3-Dihydro-1,4-benzodioxin-5-yl)-piperazine hydrochloride.

Appearance White solid

CAS # 98206-09-8

Molecular Formula C₁₂H₁₆N₂O₂HCl

Molecular Weight 256.73

Purity ≥ 98% by HPLC

Solubility H₂O (20 mg/ml)

SMILES C1CN(CCN1)C2=C3C(=CC=C2)OCCO3

InChi InChI=1S/C12H16N2O2/c1-2-10(14-6-4-13-5-7-14)12-11(3-1)15-8-9-16-12/h1-3,13H,4-9H2

InChi Key WVLHGCRWEHCIOT-UHFFFAOYSA-N

PubChem CID 65853

MDL Number MFCD06245586

Storage Conditions -20°C

Shipping Conditions Gel Pack

Usage For Research Use Only! Not For Use in Humans.

Handling Protect from air and moisture. Do not take it internally. Wear gloves and a mask when handling the product! Avoid contact by all modes of exposure.

Eltoprazine is a selective serotonin receptor agonist and antagonist that has been studied for its potential therapeutic applications in various neurological and psychiatric disorders, 5-HT1A, 5-HT1B, and 5-HT2B receptors (Kis = 40, 52, and 81 nM, respectively). Eltoprazine has shown potential in reducing aggression and impulsive behavior in certain psychiatric disorders, including intermittent explosive disorder and aggression associated with developmental disorders. It has also been investigated as a potential treatment for ADHD and Tourette syndrome.